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Synthesis of a new series of pyrazolo[1,5-a]pyrimidines as CDK2 inhibitors and anti-leukemia

Samar J. Almehmadi, Amani M.R. Alsaedi, Marwa F. Harras, Thoraya A. Farghaly

2021Bioorganic Chemistry56 citationsDOI

Topics & Concepts

ChemistryADMEIC50CytotoxicityStereochemistryPotencyPyrimidineCyclin-dependent kinase 1PharmacologyCombinatorial chemistryBiochemistryIn vitroCell cycleCellMedicineAdvanced Breast Cancer TherapiesChronic Lymphocytic Leukemia ResearchCancer-related Molecular Pathways
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