PEGylated solid lipid nanoparticles for brain delivery of lipophilic kiteplatin Pt(IV) prodrugs: An in vitro study
Ilaria Arduino, Nicoletta Depalo, Francesca Re, Roberta Dal Magro, Annamaria Panniello, Nicola Margiotta, Elisabetta Fanizza, Antonio Lopalco, Valentino Laquintana, Annalisa Cutrignelli, Angela Lopedota, Massimo Franco, Nunzio Denora
Topics & Concepts
ProdrugLipophilicitySolid lipid nanoparticlePolyethylene glycolChemistryIn vitroPEG ratioBlood–brain barrierNanoparticleAmphiphileCytotoxicityCombinatorial chemistryDrug deliveryBiophysicsStereochemistryNanotechnologyOrganic chemistryMaterials scienceBiochemistryCopolymerPolymerEconomicsCentral nervous systemBiologyNeuroscienceFinanceGold and Silver Nanoparticles Synthesis and ApplicationsNanoparticle-Based Drug DeliveryAdvanced biosensing and bioanalysis techniques