Discovery and biological evaluation of 6-aryl-4-(3,4,5-trimethoxyphenyl)quinoline derivatives with promising antitumor activities as novel colchicine-binding site inhibitors
Qianqian Xu, Yuxuan Tu, Yujing Zhang, Yutao Xiu, Zongjiang Yu, Hongfei Jiang, Chao Wang
Topics & Concepts
ChemistryQuinolineColchicineArylCombinatorial chemistryDrug discoveryBinding sitePharmacologyStereochemistryBiochemistryOrganic chemistryMedicineAlkylInternal medicineSynthesis and biological activitySynthesis and Biological EvaluationSynthesis of heterocyclic compounds