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Metabolomic Profiling and Drug Interaction Characterization Reveal Riboflavin As a Breast Cancer Resistance Protein–Specific Endogenous Biomarker That Demonstrates Prediction of Transporter Activity In Vivo

Yueping Zhang, Petia Shipkova, Bethanne M. Warrack, David M. Nelson, Linna Wang, Runlan Huo, Jian Chen, Erika Panfen, Xueqing Chen, R. Marcus Fancher, Qian Ruan, Lisa J. Christopher, Yongjun Xue, Michael Sinz, Hong Shen

2023Drug Metabolism and Disposition15 citationsDOI

Topics & Concepts

Abcg2PharmacologyIn vivoChemistryTransporterMetaboliteMetabolomicsP-glycoproteinBiomarkerPharmacokineticsATP-binding cassette transporterBiochemistryBiologyMultiple drug resistanceAntibioticsBiotechnologyGeneChromatographyDrug Transport and Resistance MechanismsPharmacological Effects and Toxicity StudiesFolate and B Vitamins Research
Metabolomic Profiling and Drug Interaction Characterization Reveal Riboflavin As a Breast Cancer Resistance Protein–Specific Endogenous Biomarker That Demonstrates Prediction of Transporter Activity In Vivo | Litcius