The Effect of Itraconazole on the Pharmacokinetics of Vepdegestrant, a PROteolysis TArgeting Chimera Estrogen Receptor Degrader, in Healthy Adult Participants
Lana Tran, Jennifer A. Winton, Kyle Matschke, Alexandre Stouffs, Kimberly C. Lee, Yuanyuan Zhang, Weiwei Tan
Topics & Concepts
MedicinePharmacokineticsItraconazolePharmacologyChimera (genetics)ProteolysisCYP3A4ReceptorEstrogen receptorEstrogenOestrogen receptorPharmacogenetics and Drug MetabolismEstrogen and related hormone effectsMenopause: Health Impacts and Treatments