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Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib

Hardik Joshi, Vijay Patil, Kalpana Tilekar, Neha Upadhyay, Vikram Gota, C. S. Ramaa

2020Bioorganic & Medicinal Chemistry Letters18 citationsDOI

Topics & Concepts

ImatinibChemistryPharmacologyIn vivoTyrosine kinaseCell growthApoptosisCyclin D1Tyrosine-kinase inhibitorIn vitroCell cycleCancer researchMyeloid leukemiaBiochemistryMedicineInternal medicineSignal transductionCancerBiologyBiotechnologyChronic Myeloid Leukemia TreatmentsQuinazolinone synthesis and applicationsPI3K/AKT/mTOR signaling in cancer
Benzylidene thiazolidinediones: Synthesis, in vitro investigations of antiproliferative mechanisms and in vivo efficacy determination in combination with Imatinib | Litcius