Schematic-portfolio of potent anti-microbial scaffolds targeting DNA gyrase: Unlocking ways to overcome resistance
Kakarla Pakeeraiah, Suvadeep Mal, Monalisa Mahapatra, Suman Kumar Mekap, Pratap Kumar Sahu, Sudhir Kumar Paidesetty
Topics & Concepts
DNA gyraseNovobiocinCiprofloxacinGatifloxacinMultiple drug resistanceDrug developmentDrug discoveryChemistryAntibioticsPharmacologyBiologyDrugMicrobiologyBiochemistryEscherichia coliGeneCancer therapeutics and mechanismsSynthesis and biological activitySynthesis and Biological Evaluation