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Medicinal chemistry updates of novel HDACs inhibitors (2020 to present)

Xingrui He, Zi Hui, Li Xu, Renren Bai, Yuan Gao, Zongcheng Wang, Tian Xie, Xiang‐Yang Ye

2021European Journal of Medicinal Chemistry76 citationsDOIOpen Access PDF

Topics & Concepts

Drug discoveryChemistryHistoneComputational biologyAcetylationHistone deacetylaseRational designPharmacologyBiochemistryBiologyGeneGeneticsHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsClick Chemistry and Applications
Medicinal chemistry updates of novel HDACs inhibitors (2020 to present) | Litcius