Discovery of novel VEGFR-2-PROTAC degraders based on the localization of lysine residues via recruiting VHL for the treatment of gastric cancer
Xingrong Wang, Shuai Wang, Hong-Xia Mu, Kai-Yan Xu, Xueting Wang, Jian-Tao Shi, Qi-Hang Cui, Liwen Zhang, Shi‐Wu Chen
Topics & Concepts
ChemistryProtein degradationProteasomeAngiogenesisCancer researchIn vitroUbiquitinCancer cellLysineApoptosisCancerBiochemistryAmino acidBiologyGeneGeneticsProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysPeptidase Inhibition and Analysis