Mining Public Domain Data to Develop Selective DYRK1A Inhibitors
Scott H. Henderson, F.J. Sorrell, James M. Bennett, Marcus T. Hanley, Sean W. Robinson, Iva Navrátilová, Jonathan M. Elkins, Simon E. Ward
Abstract
, a highly selective DYRK1A inhibitor.
Topics & Concepts
KinomeDYRK1AGSK-3KinaseCyclin-dependent kinaseDrug discoveryComputational biologyCyclin-dependent kinase 9Computer scienceBiochemistryChemistryBiologyCyclin-dependent kinase 2Protein kinase ACell cycleGeneUbiquitin and proteasome pathwaysCancer-related gene regulationNeuroblastoma Research and Treatments