Parsing structural fragments of thiazolidin-4-one based α-amylase inhibitors: A combined approach employing in vitro colorimetric screening and GA-MLR based QSAR modelling supported by molecular docking, molecular dynamics simulation and ADMET studies
Rahul Singh, Prof Parvin Kumar, Jayant Sindhu, Meena Devi, Ashwani Kumar, Sohan Lal, Devender Singh
Topics & Concepts
Quantitative structure–activity relationshipMolecular dynamicsDocking (animal)ParsingComputer scienceBiological systemMolecular modelComputational biologyChemistryArtificial intelligenceStereochemistryMachine learningComputational chemistryBiologyNursingMedicineComputational Drug Discovery MethodsEnzyme Production and CharacterizationClick Chemistry and Applications