Discovery of novel human lactate dehydrogenase inhibitors: Structure-based virtual screening studies and biological assessment
Laura Di Magno, Antonio Coluccia, M Bufano, Silvia Ripa, Giuseppe La Regina, Marianna Nalli, Fiorella Di Pastena, Gianluca Canettieri, Romano Silvestri, Luigi Frati
Topics & Concepts
ChemistryBiochemistryLactate dehydrogenaseGlycolysisCofactorCancer cellLactate dehydrogenase AOxidative phosphorylationNAD+ kinaseEffectorEnzymeCancerBiologyGeneticsCancer, Hypoxia, and MetabolismATP Synthase and ATPases ResearchBiochemical and Molecular Research