Molecular docking studies and biological evaluation of isoxazole-carboxamide derivatives as COX inhibitors and antimicrobial agents
Mohammed Hawash, Nidal Jaradat, Murad Abualhasan, Mohammed T. Qaoud, Yara Joudeh, Zeina Jaber, Majd Sawalmeh, Abdulraziq Zarour, Ahmed Mousa, Mohammed Arar
Topics & Concepts
IsoxazoleADMEChemistryDocking (animal)EnzymeStereochemistryAntimicrobialKlebsiella pneumoniaTriazoleMolecular modelIn vitroBiochemistryEscherichia coliMedicineOrganic chemistryNursingGeneSynthesis and biological activitySynthesis and Biological EvaluationInflammatory mediators and NSAID effects