Discovery of IAP-recruiting BCL-XL PROTACs as potent degraders across multiple cancer cell lines
Xuan Zhang, Yonghan He, Peiyi Zhang, Vivekananda Budamagunta, Dongwen Lv, Dinesh Thummuri, Yang Yang, Jing Pei, Yaxia Yuan, Daohong Zhou, Guangrong Zheng
Topics & Concepts
Ubiquitin ligaseChemistryUbiquitinCell cultureDNA ligaseCereblonCancer researchBiologyBiochemistryGeneticsDNAGeneProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsPeptidase Inhibition and Analysis