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Disposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating Metabolites

Takashi Ueno, T. Ishida, Jagadeesh Aluri, Michiyuki Suzuki, Carsten T. Beuckmann, Takaaki Kameyama, Shoji Asakura, Kazutomi Kusano

2020Drug Metabolism and Disposition24 citationsDOIOpen Access PDF

Topics & Concepts

MetaboliteGlucuronidationPharmacologyUrineMetabolismPharmacokineticsChemistryFecesAntagonistReceptorBiologyBiochemistryIn vitroMicrosomePaleontologySleep and Wakefulness ResearchSleep and related disordersCircadian rhythm and melatonin
Disposition and Metabolism of [14C]Lemborexant in Healthy Human Subjects and Characterization of Its Circulating Metabolites | Litcius