Discovery of novel urea-diarylpyrazole hybrids as dual COX-2/sEH inhibitors with improved anti-inflammatory activity and highly reduced cardiovascular risks
Ahmed H. Abdelazeem, Asmaa G. Safi El-Din, Maha M. Abdel‐Fattah, Noha H. Amin, Samir M. El‐Moghazy, Mohammed T. El‐Saadi
Topics & Concepts
ChemistryCelecoxibPharmacologyLactate dehydrogenaseCreatine kinaseIn vivoProstacyclinEnzymeBiochemistryMedicineBiotechnologyBiologyEicosanoids and Hypertension PharmacologyInflammatory mediators and NSAID effectsSynthesis and biological activity