Design, synthesis and evaluation of novel monoamine oxidase B (MAO-B) inhibitors with improved pharmacokinetic properties for Parkinson's disease
Chao Yi, Xinchang Liu, Kangzhi Chen, Haiping Liang, Chuanfei Jin
Topics & Concepts
BenzofuranChemistryPyrrolidineMonoamine oxidaseCarboxamidePharmacologyMPTPPharmacokineticsMonoamine oxidase BStereochemistryMoietyDopamineBiochemistryInternal medicineEnzymeDopaminergicMedicineParkinson's Disease Mechanisms and TreatmentsCholinesterase and Neurodegenerative DiseasesAlzheimer's disease research and treatments