Computational exploration and experimental validation to identify a dual inhibitor of cholinesterase and amyloid-beta for the treatment of Alzheimer’s disease
Manish Tripathi, Piyoosh Sharma, Avanish Tripathi, Prabhash Nath Tripathi, Pavan Srivastava, Ankit Seth, Sushant K. Shrivastava
Topics & Concepts
CholinesteraseDocking (animal)Amyloid betaThioflavinNeuroprotectionIC50Virtual screeningAchéChemistryAcetylcholinesteraseButyrylcholinesterasePharmacologyIn vitroEnzymeBiochemistryAlzheimer's diseaseDiseaseMedicineInternal medicineDrug discoveryPeptideNursingCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsNicotinic Acetylcholine Receptors Study