Discovery of novel selenium-containing azole derivatives as antifungal agents by exploiting the hydrophobic cleft of CYP51
Hang Xu, Yanhua Mou, Mengbi Guo, Rui Zhang, Zhong-zuo Yan, Ran An, Xin Wang, Xin Su, Zhuang Hou, Chun Guo
Topics & Concepts
ChemistryAntifungalFluconazoleHemolysisIn vivoDocking (animal)StereochemistryMicrobiologyBiologyMedicineImmunologyBiotechnologyNursingAntifungal resistance and susceptibilitySynthesis and Biological EvaluationOrganoselenium and organotellurium chemistry