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Contribution of UGT Enzymes to Human Drug Metabolism Stereoselectivity: A Case Study of Medetomidine, RO5263397, Propranolol, and Testosterone

Nicolò Milani, NaHong Qiu, Stephen Fowler

2022Drug Metabolism and Disposition15 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryStereoselectivityGlucuronidationEnzymeDrug metabolismGlucuronosyltransferaseCytochrome P450MetabolismBiochemistryMicrosomeCatalysisPharmacogenetics and Drug MetabolismAnalytical Chemistry and ChromatographyDrug Transport and Resistance Mechanisms
Contribution of UGT Enzymes to Human Drug Metabolism Stereoselectivity: A Case Study of Medetomidine, RO5263397, Propranolol, and Testosterone | Litcius