Development of potent inhibitors of the human microsomal epoxide hydrolase
Bogdan Barnych, Nalin Singh, Sophie Négrel, Yue Zhang, Damien Magis, Capucine Roux, Xiude Hua, Zhewen Ding, Christophe Morisseau, Dean J. Tantillo, Justin B. Siegel, Bruce D. Hammock
Topics & Concepts
ChemistryEpoxide hydrolasePharmacophoreMicrosomal epoxide hydrolaseEpoxide hydrolase 2EnzymeAcetamideStereochemistryDocking (animal)BiochemistryAmideHydrolaseHomology modelingMicrosomeOrganic chemistryNursingMedicineEicosanoids and Hypertension PharmacologyPharmacogenetics and Drug MetabolismBiochemical Acid Research Studies