Subtype-selective mechanisms of negative allosteric modulators binding to group I metabotropic glutamate receptors
Tingting Fu, Gao Tu, Ping Meng, Guoxun Zheng, Fengyuan Yang, H. J. Yang, Yang Zhang, Xiaojun Yao, Weiwei Xue, Feng Zhu
Topics & Concepts
Metabotropic glutamate receptorAllosteric regulationMetabotropic receptorMetabotropic glutamate receptor 1Metabotropic glutamate receptor 2Metabotropic glutamate receptor 5Docking (animal)Computational biologyGlutamate receptorChemistryReceptorBinding siteClass C GPCRStereochemistryBiologyBiochemistryMedicineNursingReceptor Mechanisms and SignalingNeuroscience and Neuropharmacology ResearchNicotinic Acetylcholine Receptors Study