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Synthesis and biological evaluation of new 2‑substituted‑4‑amino-quinolines and -quinazoline as potential antifungal agents

Tianhong Qin, Jianchuan Liu, Jinyuan Zhang, Lin-Xiu Tang, Yanni Ma, Yang Rui

2022Bioorganic & Medicinal Chemistry Letters35 citationsDOI

Topics & Concepts

QuinazolineChemistryAntifungalAntifungal drugAmine gas treatingCombinatorial chemistryStereochemistryBiological activityPotencyCarbon-13 NMRStructure–activity relationshipProton NMRMinimum inhibitory concentrationIn vitroBiochemistryOrganic chemistryMicrobiologyBiologyQuinazolinone synthesis and applicationsSynthesis and biological activitySynthesis and Biological Evaluation
Synthesis and biological evaluation of new 2‑substituted‑4‑amino-quinolines and -quinazoline as potential antifungal agents | Litcius