Ball-milling synthesis of sulfonyl quinolines <i>via</i> coupling of haloquinolines with sulfonic acids
Xiaowen Liu, Jia-Qian Wang, Hui Ma, Qi Zhu, Long‐Yong Xie
Abstract
A practical and environment-friendly methodology for the construction of sulfonyl quinolines through ball milling promoted coupling of haloquinolines with sulfonic acid under metal-, base-, solvent- and additive-free conditions was developed.
Topics & Concepts
SulfonylBall millSulfonic acidChemistrySolventCoupling (piping)Organic chemistryCombinatorial chemistryMaterials scienceMetallurgyAlkylSulfur-Based Synthesis TechniquesPhenothiazines and Benzothiazines Synthesis and ActivitiesCatalytic C–H Functionalization Methods