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Synthesis of Novel G Factor or Chloroquine-Artemisinin Hybrids and Conjugates with Potent Antiplasmodial Activity

Dionissia A. Pepe, Dimitra Toumpa, Christiane André‐Barrès, Christophe Menendez, Elisabeth Mouray, Michel Baltas, Philippe Grellier, Dionissios Papaioannou, Constantinos M. Athanassopoulos

2020ACS Medicinal Chemistry Letters29 citationsDOIOpen Access PDF

Abstract

of Hsd.

Topics & Concepts

ConjugateArtemisininPlasmodium falciparumChloroquineSpermidineIC50ChemistryIn vitroStereochemistryBiologyBiochemistryMalariaImmunologyEnzymeMathematicsMathematical analysisMalaria Research and ControlPhenothiazines and Benzothiazines Synthesis and ActivitiesTrypanosoma species research and implications
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