Litcius/Paper detail

Synthesis, biochemical and computational evaluations of novel bis-acylhydrazones of 2,2′-(1,1′-biphenyl)-4,4′-diylbis(oxy))di(acetohydrazide) as dual cholinesterase inhibitors

Muhammad Ibrahim, Sobia Ahsan Halim, Abdul Latif, Manzoor Ahmad, Sajid Ali, Samee Ullah, Asaad Khalid, Ashraf N. Abdalla, Ajmal Khan, Ahmed Al‐Harrasi, Mumtaz Ali, Mumtaz Ali

2024Bioorganic Chemistry11 citationsDOI

Topics & Concepts

ChemistryButyrylcholinesteraseAcetylcholinesteraseCholinesteraseIC50StereochemistryAchéHydrazine (antidepressant)EnzymeMedicinal chemistryIn vitroCombinatorial chemistryOrganic chemistryBiochemistryPharmacologyMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsEnzyme function and inhibition