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Ruthenium-Catalyzed Asymmetric <i>N</i>-Acyl Nitrene Transfer Reaction: Imidation of Sulfide

Masaki Yoshitake, Hiroki Hayashi, Tatsuya Uchida

2020Organic Letters64 citationsDOI

Abstract

-acyl nitrene intermediates without any activation via heating or UV irradiation, or transfer generating nitrene intermediates to the sulfur atom of sulfides with good to excellent enantioselectivities (≤98% ee) without diazene and isocyanate contamination.

Topics & Concepts

NitreneChemistryRutheniumCatalysisSulfideTransfer (computing)Combinatorial chemistryPhotochemistryOrganic chemistryMedicinal chemistryParallel computingComputer scienceSynthesis and Catalytic ReactionsCatalytic C–H Functionalization MethodsAsymmetric Hydrogenation and Catalysis
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