Design, synthesis, biological assessment, and in-Silico studies of 1,2,4-triazolo[1,5-a]pyrimidine derivatives as tubulin polymerization inhibitors
Heba S. Mohamed, Noha H. Amin, Mohammed T. El‐Saadi, Hamdy M. Abdel‐Rahman
Topics & Concepts
ChemistryTubulinPyrimidineCombretastatinStereochemistryDocking (animal)Cell cycleMicrotubuleMicrotubule polymerizationIC50PolymerizationApoptosisColchicineCell cycle checkpointIn vitroBiochemistryCell biologyBiologyOrganic chemistryMedicinePolymerGeneticsNursingSynthesis and biological activityClick Chemistry and ApplicationsSynthesis and Characterization of Heterocyclic Compounds