Litcius/Paper detail

Discovery of coumarin derivatives as potent and selective cyclin-dependent kinase 9 (CDK9) inhibitors with high antitumour activity

Junyu Xu, Hongmei Li, Xinren Wang, Jianhang Huang, Shuwen Li, Chenhe Liu, Ruinan Dong, Gaoyuan Zhu, Chunqi Duan, Fei Jiang, Yanmin Zhang, Yuqin Zhu, Tianyi Zhang, Yadong Chen, Weifang Tang, Tao Lu

2020European Journal of Medicinal Chemistry42 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryCoumarinCyclin-dependent kinaseSelectivityhERGBromodomainStereochemistryPharmacologyBiochemistryBiophysicsApoptosisCell cycleAcetylationPotassium channelMedicineGeneBiologyCatalysisOrganic chemistryCancer-related Molecular PathwaysAcute Myeloid Leukemia ResearchProtein Degradation and Inhibitors