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Synthesis and evaluation of 1,2,4-oxadiazole derivatives as potential anti-inflammatory agents by inhibiting NF-κB signaling pathway in LPS-stimulated RAW 264.7 cells

Yuying Zhang, Qianqian Zhang, Juan Zhang, Jiali Song, Jiacheng Li, Ke Han, Jintian Huang, Cheng‐Shi Jiang, Hua Zhang

2020Bioorganic & Medicinal Chemistry Letters23 citationsDOI

Topics & Concepts

ChemistryNF-κBBlotAnti-inflammatoryLuciferasePhosphorylationOxadiazoleLipopolysaccharideSignal transductionIκBαPharmacologyBiochemistryTransfectionImmunologyBiologyGeneOrganic chemistryNF-κB Signaling PathwaysCytokine Signaling Pathways and InteractionsSynthesis and biological activity
Synthesis and evaluation of 1,2,4-oxadiazole derivatives as potential anti-inflammatory agents by inhibiting NF-κB signaling pathway in LPS-stimulated RAW 264.7 cells | Litcius