Novel potent (dihydro)benzofuranyl piperazines as human histamine receptor ligands – Functional characterization and modeling studies on H3 and H4 receptors
Michelle Fidelis Corrêa, André L. Balico-Silva, Dóra Kiss, Gustavo Ariel Borges Fernandes, Jhonatan Christian Maraschin, Lucas T. Parreiras‐e‐Silva, Marina T. Varela, Sarah C. Simões, Michel Bouvier, György M. Keserű, Cláudio M. Costa-Neto, João Paulo S. Fernandes
Topics & Concepts
ChemistryHistamineHistamine H3 receptorStereochemistryAgonistReceptorPharmacophoreDocking (animal)Histamine H4 receptorPartial agonistBenzofuranPharmacologyHistamine H2 receptorBiochemistryAntagonistNursingMedicineMast cells and histamineReceptor Mechanisms and SignalingChemical Synthesis and Analysis