Design, synthesis, in vitro, and in silico studies of new thiadiazol derivatives as promising VEGFR-2 inhibitors and apoptosis inducers
Hazem A. Mahdy, Hazem Elkady, Walid E. Elgammal, Eslam B. Elkaeed, Aisha A. Alsfouk, Ibrahim M. Ibrahim, Dalal Z. Husein, Mohamed A. Elkady, Ahmed M. Metwaly, Ibrahim H. Eissa
Topics & Concepts
ChemistryIn silicoApoptosisIn vitroCell cycleIC50SorafenibDocking (animal)StereochemistryInducerCell cultureCell cycle checkpointCancer cellPharmacologyBiochemistryCancer researchCancerInternal medicineMedicineGeneticsNursingBiologyHepatocellular carcinomaGeneSynthesis and biological activityPI3K/AKT/mTOR signaling in cancerClick Chemistry and Applications