EGFR-targeted prodrug activation using bioorthogonal alkene-azide click-and-release chemistry
Jessica M. Fairhall, Júlia Constantino Camilli, Blake Gibson, Sarah Hook, Allan B. Gamble
Topics & Concepts
Bioorthogonal chemistryProdrugChemistryClick chemistryDoxorubicinCetuximabEpidermal growth factor receptorCancer researchCombinatorial chemistryBiochemistryMonoclonal antibodyAntibodyReceptorChemotherapyImmunologyBiologyMedicineInternal medicineClick Chemistry and ApplicationsMonoclonal and Polyclonal Antibodies ResearchProtein Degradation and Inhibitors