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What makes a good fragment in fragment-based drug discovery?

Zenon Konteatis

2021Expert Opinion on Drug Discovery30 citationsDOIOpen Access PDF

Abstract

Over the past 25 years, fragment-based drug discovery (FBDD) has emerged as a highly successful, complementary approach to high-throughput screening (HTS) to identify quality leads for optimization...

Topics & Concepts

Fragment (logic)Drug discoveryComputational biologyComputer scienceDrugBiologyBioinformaticsPharmacologyAlgorithmComputational Drug Discovery MethodsMicrobial Natural Products and BiosynthesisBioinformatics and Genomic Networks
What makes a good fragment in fragment-based drug discovery? | Litcius