Synthesis, biological evaluation and action mechanism of 7H-[1,2,4] triazolo [3,4-b] [1,3,4] thiadiazine-phenylhydrazone derivatives as α-glucosidase inhibitors
Qianqian Feng, Jinfeng Zhang, Shuang Luo, Yong Huang, Zhiyun Peng, Guangcheng Wang
Topics & Concepts
ChemistryAcarboseStereochemistryIC50In vivoDocking (animal)CytotoxicityMechanism of actionCircular dichroismPostprandialProton NMRActive siteCarbon-13 NMREnzymePotencyIn vitroBiochemistryMedicineBiologyEndocrinologyNursingInsulinBiotechnologySynthesis and biological activitySynthesis and Characterization of Heterocyclic CompoundsClick Chemistry and Applications