Degraders: The Ultimate Weapon Against Amplified Driver Kinases in Cancer
Pedro Torres‐Ayuso, John Brognard
Topics & Concepts
KinaseCarcinogenesisBiologyProtein-Serine-Threonine KinasesCell biologyGeneCancer researchGeneticsProtein kinase AProtein Degradation and InhibitorsUbiquitin and proteasome pathwaysClick Chemistry and Applications