Functional assessment of the effects of CYP3A4 variants on acalabrutinib metabolism in vitro
Mingming Han, Jianchang Qian, Zhize Ye, Ren-ai Xu, Daoxing Chen, Saili Xie, Jianping Cai, Guoxin Hu
Topics & Concepts
CYP3A4ChemistryKetoconazoleMicrosomeMetabolismEnzymePharmacologyCytochrome P450BiochemistryBiologyAntifungalMicrobiologyChronic Lymphocytic Leukemia ResearchMyeloproliferative Neoplasms: Diagnosis and TreatmentChronic Myeloid Leukemia Treatments