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Palladium-catalyzed synthesis of spirooxindoles and [3,4]-fused oxindoles from alkene-tethered carbamoyl chlorides

Fang Yang, Wan Sun, Haifang Meng, Mengjia Chen, Chen Chen, Bolin Zhu

2020Organic Chemistry Frontiers24 citationsDOI

Abstract

We disclosed an efficient Pd-catalyzed domino reaction for the synthesis of spirooxindoles and [3,4]-fused oxindoles from alkene-tethered carbamoyl chlorides.

Topics & Concepts

ChemistryAlkeneDominoCatalysisPalladiumCombinatorial chemistryCascade reactionOrganic chemistryCatalytic C–H Functionalization MethodsSynthesis and Catalytic ReactionsCyclopropane Reaction Mechanisms
Palladium-catalyzed synthesis of spirooxindoles and [3,4]-fused oxindoles from alkene-tethered carbamoyl chlorides | Litcius