Litcius/Paper detail

The influence of calculated physicochemical properties of compounds on their ADMET profiles

Shifan Ma, Mark McGann, Istvan Enyedy

2021Bioorganic & Medicinal Chemistry Letters16 citationsDOI

Topics & Concepts

hERGChemistryBioavailabilityEffluxPharmacokineticsLipophilicityMicrosomeStereochemistryPharmacologyBiophysicsBiochemistryIn vitroPotassium channelMedicineBiologyReceptor Mechanisms and SignalingDrug Transport and Resistance MechanismsComputational Drug Discovery Methods