Novel antiproliferative agents bearing morpholinopyrimidine scaffold as PI3K inhibitors and apoptosis inducers; design, synthesis and molecular docking
Amira A. Helwa, Nehad M. El‐Dydamony, Rasha Ali Radwan, Sahar M. Abdelraouf, Rana M. Abdelnaby
Topics & Concepts
ChemistryDocking (animal)ApoptosisAnnexinIC50In vitroCytotoxic T cellCytotoxicityCell cyclePI3K/AKT/mTOR pathwayCell cultureGrowth inhibitionStereochemistryBiochemistryBiologyGeneticsMedicineNursingBiochemical and Molecular ResearchPI3K/AKT/mTOR signaling in cancerCancer therapeutics and mechanisms