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Natural phenolics as multitarget antimicrobials for food preservation: mechanisms of action

Lei Zhao, Ya Zhou, Weiguo Yue, Qingshan Shen, Jingxuan Ke, Yanli Ma, Lifang Zhang, Hua Bian

2025Food Chemistry X20 citationsDOIOpen Access PDF

Abstract

Natural phenolics are emerging as promising clean-label antimicrobials, yet evidence for their multitarget mechanisms remains scattered. This review synthesizes 158 studies (2013–2025) on Escherichia coli , Staphylococcus aureus , and related pathogens. Three converging antibacterial targets are identified: ROS generation (72 % of phenolics), membrane disruption (58 %), and DNA interaction (41 %). Compounds such as bisdemethoxycurcumin, gallic acid, thymol, and Epigallocatechin gallate (EGCG) act across all targets, reducing bacterial counts by up to 4 log CFU/mL at ≤2 × MIC. A cascade mechanism is proposed: ROS triggers lipid peroxidation, weakening membranes, enhancing phenolic uptake, and accelerating DNA damage. Food matrix factors (pH, fat, water activity, microbiota) can suppress efficacy by up to 90 %. Emerging delivery strategies—nanoemulsions, biopolymer capsules, and active films—partially restore function. This review integrates molecular insights with food system data, offering a practical framework for designing robust phenolic-based antimicrobials. • Natural phenolics disrupt bacteria via ROS, membrane damage, and DNA binding. • A cascade model explains how multitarget synergy enhances antimicrobial efficacy. • Experimental data verify BDMC's DNA interaction and oxidative membrane stress. • Food matrix interference and delivery strategies are critically reviewed. • Insights guide the clean-label design of phenolic-based food preservatives.

Topics & Concepts

ChemistryAntimicrobialGallic acidPolyphenolEpigallocatechin gallateGallateAction (physics)Mechanism (biology)Mechanism of actionBiopolymerGreen teaDNANatural (archaeology)Food productsBiochemistryNatural compoundFood scienceAnti-Infective AgentsBiologyComputational biologyBiotechnologyEpicatechin gallateHealth benefitsTraditional medicineFlavonoidDNA damageBiochemical engineeringTranscriptomeBiological activityCatechinPhytochemicals and Antioxidant ActivitiesEssential Oils and Antimicrobial ActivityBee Products Chemical Analysis
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