Evaluation of novel 2-(quinoline-2-ylthio)acetamide derivatives linked to diphenyl-imidazole as α-glucosidase inhibitors: Insights from in silico, in vitro, and in vivo studies on their anti-diabetic properties
Minoo Khalili Ghomi, Milad Noori, Maryam Mirahmad, Aida Iraji, Ahmad Shahir Sadr, Navid Dastyafteh, Pooria Asili, Mahdi Gholami, Shahrzad Javanshir, Maryam Lotfi, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Mehdi Asadi, Ensieh Nasli‐Esfahani, Mahdie Palimi, Bagher Larijani, Mohammad Hadi Meshkatalsadat, Mohammad Mahdavi
Topics & Concepts
AcarboseChemistryQuinolineIn vivoAcetamideIn silicoImidazoleIn vitroEnzymeIC50PharmacologyBiochemistryDocking (animal)StereochemistryPotencyBiologyOrganic chemistryMedicineBiotechnologyGeneNursingNatural Antidiabetic Agents StudiesComputational Drug Discovery MethodsSynthesis and biological activity