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Rational drug design of benzothiazole-based derivatives as potent signal transducer and activator of transcription 3 (STAT3) signaling pathway inhibitors

Dingding Gao, Nan Jin, Yixian Fu, Yueyue Zhu, Yujie Wang, Ting Wang, Yuehong Chen, Mingming Zhang, Qiang Xiao, Min Huang, Yingxia Li

2021European Journal of Medicinal Chemistry28 citationsDOIOpen Access PDF

Topics & Concepts

STAT3ChemistrySTAT proteinBenzothiazoleSignal transductionApoptosisPhosphorylationCancer researchBiochemistryBiologyCytokine Signaling Pathways and InteractionsCancer Mechanisms and TherapyHER2/EGFR in Cancer Research
Rational drug design of benzothiazole-based derivatives as potent signal transducer and activator of transcription 3 (STAT3) signaling pathway inhibitors | Litcius