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Development of High-Throughput Assays for Evaluation of Hematopoietic Progenitor Kinase 1 Inhibitors

Brian M. Lacey, Zangwei Xu, Xiaomei Chai, Jason Laskey, Xavier Fradera, Payal Mittal, Sasmita Mishra, Jennifer Piesvaux, P Saradjian, Lynsey Shaffer, Galya Vassileva, Catherine Gerdt, Yun Wang, Heidi M. Ferguson, Dustin Smith, Jeanine Ballard, Steven B. Wells, Rishabh Jain, U. Müeller, George H. Addona, Ilona Kariv, Joey L. Methot, Mark Bittinger, Sheila Ranganath, Robbie L. McLeod, Alexander Pasternak, J. Richard Miller, Haiyan Xu

2020SLAS DISCOVERY28 citationsDOIOpen Access PDF

Topics & Concepts

KinaseCell biologyBiologyProgenitor cellProtein kinase AMolecular biologyCyclin-dependent kinase 9Mitogen-activated protein kinase kinaseChemistryBiochemistryStem cellMelanoma and MAPK PathwaysImmune cells in cancerCytokine Signaling Pathways and Interactions
Development of High-Throughput Assays for Evaluation of Hematopoietic Progenitor Kinase 1 Inhibitors | Litcius