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Tuning sterol extraction kinetics yields a renal-sparing polyene antifungal

Arun Maji, Corinne P. Soutar, Jiabao Zhang, Agnieszka Lewandowska, Brice E. Uno, Yan Su, Yogesh G. Shelke, Ganesh M. Murhade, Evgeny Nimerovsky, Collin G. Borcik, Andres S. Arango, Justin Lange, J. Marin-Toledo, Yinghuan Lyu, Keith Bailey, Patrick J. Roady, Jordan T. Holler, Anuj Khandelwal, Anna M. SantaMaria, Hiram Sánchez, Praveen R. Juvvadi, Gina Johns, Michael J. Hageman, Joanna Krise, Teclegiorgis Gebremariam, Eman G. Youssef, Ken Bartizal, Kieren A. Marr, William J. Steinbach, Ashraf S. Ibrahim, Thomas F. Patterson, Nathan P. Wiederhold, David R. Andes, Taras V. Pogorelov, Charles D. Schwieters, Timothy M. Fan, Chad M. Rienstra, Martin D. Burke

2023Nature98 citationsDOIOpen Access PDF

Topics & Concepts

PolyeneErgosterolAmphotericin BSterolChemistryBiochemistryBiologyMicrobiologyPharmacologyAntifungalCholesterolCholinesterase and Neurodegenerative DiseasesAntifungal resistance and susceptibilityIonic liquids properties and applications
Tuning sterol extraction kinetics yields a renal-sparing polyene antifungal | Litcius