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Targeting breast cancer resistance protein (BCRP/ABCG2): Functional inhibitors and expression modulators

Ingrid Fátima Zattoni, Letícia Carani Delabio, Júlia de Paula Dutra, Diogo Henrique Kita, Gustavo Scheiffer, Marina Hembecker, Giovana da Silva Pereira, Vivian Rotuno Moure, Gláucio Valdameri

2022European Journal of Medicinal Chemistry79 citationsDOIOpen Access PDF

Topics & Concepts

Abcg2Breast cancerMultiple drug resistanceCancerChemistryCancer stem cellMechanism (biology)Cancer researchPharmacologyATP-binding cassette transporterDrug resistanceTransporterEffluxComputational biologyBiologyMedicineBiochemistryInternal medicineGeneGeneticsPhilosophyEpistemologyDrug Transport and Resistance MechanismsCancer therapeutics and mechanismsRNA Interference and Gene Delivery
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