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Recent advances in developing degraders & inhibitors of lysine methyltransferases

Julia Velez, H. Ümit Kanıskan, Jian Jin

2023Current Opinion in Chemical Biology10 citationsDOIOpen Access PDF

Topics & Concepts

MethyltransferaseProteolysisLysineDrug discoveryComputational biologyBiologyEnzymeBiochemistryMethylationAmino acidDNAProtein Degradation and InhibitorsCancer-related gene regulationEpigenetics and DNA Methylation
Recent advances in developing degraders & inhibitors of lysine methyltransferases | Litcius