Design, synthesis and biological evaluation of novel fluoro-substituted benzimidazole derivatives with anti-hypertension activities
Zhuo Wu, Ming-Bao Xia, D. Bertsetseg, Yanhui Wang, Xiaolu Bao, Weibo Zhu, Tao-Xu, Pei-Ran Chen, Hesheng Tang, Yi‐Jia Yan, Zhilong Chen
Topics & Concepts
BenzimidazoleChemistryLosartanTelmisartanAngiotensin II receptor type 1PharmacologyBlood pressureAngiotensin IIAntihypertensive drugBiological activityAngiotensin receptorReceptorCombinatorial chemistryStereochemistryBiochemistryInternal medicineOrganic chemistryIn vitroMedicineReceptor Mechanisms and SignalingComputational Drug Discovery MethodsSynthesis and Catalytic Reactions