In silico Druggability Assessment of the NUDIX Hydrolase Protein Family as a Workflow for Target Prioritization
Maurice Michel, Evert Homan, Elisée Wiita, Kia Pedersen, Ingrid Almlöf, Anna‐Lena Gustavsson, Thomas Lundbäck, Thomas Helleday, Ulrika Warpman Berglund
Abstract
druggability assessment is applicable as a standalone method for decision on target prioritization and exclusion in future screening campaigns.
Topics & Concepts
DruggabilityIn silicoWorkflowComputer scienceDrug discoveryComputational biologyDocking (animal)PrioritizationBioinformaticsBiologyDatabaseEngineeringGeneticsMedicineGeneNursingManagement scienceBiochemical and Molecular ResearchEnzyme Structure and FunctionATP Synthase and ATPases Research