Identification of thiophene-benzenesulfonamide derivatives for the treatment of multidrug-resistant tuberculosis
Rongfei Qin, Pengxu Wang, Bin Wang, Lei Fu, Sarah M. Batt, Gurdyal S. Besra, Chengwei Wu, Yanan Wang, Haihong Huang, Yu Lu, Gang Li
Topics & Concepts
ChemistryAntimycobacterialDruggabilityLead compoundCytotoxicityDocking (animal)In vivoPharmacologyStructure–activity relationshipDrugBenzothiophenehERGIC50TuberculosisThiopheneMycobacterium tuberculosisStereochemistryIn vitroBiochemistryMedicineNursingGeneEndocrinologyBiotechnologyOrganic chemistryBiologyPotassium channelPathologyTuberculosis Research and EpidemiologyCancer therapeutics and mechanismsComputational Drug Discovery Methods